SCHEMBL6870352

SCHEMBL6870352

CN1CCN(C)C(c2nc3c(OC(N)=O)cccc3[nH]2)C1

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.72
PARP2 Q9UGN5 1/20 0.41
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5620255 0.84 PARP1 (1.00) PARP1PARP2
Hydrochloric Acid SCHEMBL18614474 0.83 PARP1 (0.98) PARP1PARP2
SCHEMBL6872852 0.82 PARP1 (0.72) PARP1PARP2
SCHEMBL6872354 0.81 PARP1 (0.70) PARP1PARP2
SCHEMBL6874969 0.77 PARP1 (0.51) PARP1
SCHEMBL6869690 0.76 PARP1 (0.62) PARP1PARP2
SCHEMBL6873574 0.76 PARP1 (0.73) PARP1PARP2
SCHEMBL1298068 0.76 PARP1 (0.64) PARP1PARP2
SCHEMBL6870155 0.76 PARP1 (0.62) PARP1PARP2
SCHEMBL6873107 0.75 PARP1 (0.71) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed