SCHEMBL6870679

SCHEMBL6870679

Nc1cc(C(=O)NCc2ccccc2Br)cc2nc(-c3ccc(Br)o3)nn12

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.59
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871407 0.91 ADORA2A (0.48) ADORA2AKMT2AALDH1A1LMNA
SCHEMBL6871493 0.89 ADORA2A (0.66) ADORA2A
SCHEMBL6871219 0.87 ADORA2A (0.56) ADORA2AKMT2A
SCHEMBL6871885 0.86 KMT2A (0.43) ADORA2AKMT2AALDH1A1LMNA
SCHEMBL6870074 0.85 KMT2A (0.48) ADORA2AKMT2AALDH1A1LMNA
SCHEMBL6863192 0.84 ADORA2A (0.71) ADORA2A
SCHEMBL6869214 0.83 KMT2A (0.46) ADORA2AKMT2AALDH1A1LMNA
SCHEMBL6867203 0.82 ADORA2A (0.54) ADORA2AKMT2A
SCHEMBL6870707 0.82 KMT2A (0.43) ADORA2AKMT2AALDH1A1LMNA
SCHEMBL6869437 0.82 KMT2A (0.47) ADORA2AKMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed