SCHEMBL687121

SCHEMBL687121

O=C(O)C[C@H](NC(=O)Nc1c(O)ccn(Cc2ccccc2Cl)c1=O)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.46
PTGER3 P43115 11/20 0.41
WDR5 P61964 1/20 0.39
THRB P10828 1/20 0.38
CYP1A2 P05177 1/20 0.38
SLC16A3 O15427 1/20 0.38
SLC16A1 P53985 1/20 0.38
MCTS1 Q9ULC4 1/20 0.38
CHRM5 P08912 1/20 0.37
MMP12 P39900 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGAV P06756 1/20 0.37
ITGB5 P18084 1/20 0.37
ITGB6 P18564 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688164 0.94 MAPT (0.41) MAPTPTGER3THRBCYP1A2KDM4E
SCHEMBL688306 0.92 MAPT (0.51) MAPTPTGER3THRBMMP12KDM4E
SCHEMBL688178 0.92 PTGER3 (0.42) MAPTPTGER3CYP1A2KDM4EALDH1A1
SCHEMBL687117 0.90 PTGER3 (0.52) MAPTPTGER3CYP1A2KDM4EALDH1A1
SCHEMBL27741944 0.89 CTSA (0.47) MAPTPTGER3WDR5THRBKDM4E
SCHEMBL687768 0.89 CTSA (0.47) MAPTPTGER3WDR5THRBKDM4E
SCHEMBL687597 0.89 PTGER3 (0.46) PTGER3CYP1A2SLC16A3SLC16A1MCTS1
SCHEMBL687654 0.88 PTGER3 (0.43) MAPTPTGER3CYP1A2KDM4EALDH1A1
SCHEMBL686873 0.88 PTGER3 (0.49) PTGER3CYP1A2KDM4EALDH1A1MAPK1
SCHEMBL687152 0.88 PTGER3 (0.48) PTGER3CYP1A2KDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed