SCHEMBL6872077

SCHEMBL6872077

COC(=O)c1cc(N)n2nc(-c3nccs3)nc2c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 13/20 0.42
DHFR P00374 1/20 0.41
ALDH1A1 P00352 2/20 0.39
PPARG P37231 1/20 0.39
MAPK10 P53779 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
HPGD P15428 2/20 0.38
ADORA2B P29275 1/20 0.37
ADORA1 P30542 1/20 0.37
SYK P43405 1/20 0.36
MAPT P10636 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863122 0.85 ADORA2A (0.45) ADORA2AHPGDADORA2BADORA1
SCHEMBL6871432 0.83 ADORA2A (0.40) ADORA2AALDH1A1KMT2AHPGDADORA2B
SCHEMBL6868365 0.81 ADORA2A (0.44) ADORA2AALDH1A1NPSR1RXFP1HPGD
SCHEMBL6871915 0.81 ADORA2A (0.40) ADORA2AHPGDADORA2BADORA1
SCHEMBL6871350 0.81 ADORA2A (0.41) ADORA2AADORA2BADORA1
SCHEMBL6863143 0.81 ADORA2A (0.58) ADORA2AHPGDADORA2BADORA1
SCHEMBL6867623 0.81 F2 (0.43) ADORA2AALDH1A1KMT2AHPGDADORA2B
SCHEMBL6871431 0.81 ADORA2A (0.48) ADORA2AALDH1A1KMT2AADORA2BADORA1
SCHEMBL6871970 0.81 ADORA2A (0.43) ADORA2AHPGDMAPT
SCHEMBL6870319 0.80 ADORA2A (0.49) ADORA2AHPGDADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed