SCHEMBL6876823

SCHEMBL6876823

COCC1CCCN1C(=O)c1cc(N)c2nc(-c3ccccc3)nn2c1

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.71
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
PDE4B Q07343 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12923689 1.00 ADORA2A (0.71) ADORA2ANPC1RAB9AMEN1KMT2A
SCHEMBL6885468 1.00 ADORA2A (0.71) ADORA2ANPC1RAB9AMEN1KMT2A
SCHEMBL990485 0.86 ADORA2A (0.75) ADORA2A
SCHEMBL990483 0.86 ADORA2A (0.75) ADORA2A
SCHEMBL18269267 0.86 ADORA2A (0.67) ADORA2ANPC1RAB9A
SCHEMBL6884053 0.86 ADORA2A (0.67) ADORA2ANPC1RAB9A
SCHEMBL18269264 0.86 ADORA2A (0.75) ADORA2A
SCHEMBL6884049 0.86 ADORA2A (0.67) ADORA2ANPC1RAB9A
SCHEMBL6886980 0.85 ADORA2A (0.69) ADORA2AMEN1KMT2A
SCHEMBL6879384 0.85 ADORA2A (0.68) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6689790-B2 8-AMINO-6-AMIDO-SUBSTITUTED-(1,2,4)TRIAZOLO(1,5-A)PYRIDINES; ADENOSINE RECEPTOR MODULATERS HOFFMANN-LA ROCHE INC. 2004-02-10 US disclosed