SCHEMBL6879426

SCHEMBL6879426

Cc1cc(C(=O)N[C@H]2CC[C@@H](Nc3nccc(N(C)C)n3)CC2)c(C(F)(F)F)o1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 18/20 0.50
ADRA2A P08913 9/20 0.50
HRH1 P35367 7/20 0.50
ADRA1A P35348 5/20 0.50
HTR2B P41595 7/20 0.45
CNR1 P21554 1/20 0.44
KCNH2 Q12809 1/20 0.44
AURKB Q96GD4 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HTR1A P08908 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6879429 1.00 MCHR1 (0.50) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL6880709 0.89 MCHR1 (0.51) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL6880700 0.89 MCHR1 (0.51) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL6468011 0.88 NPC1 (0.56) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL6468023 0.88 NPC1 (0.56) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL6867462 0.86 MCHR1 (0.45) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL6868121 0.85 MCHR1 (0.49) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL6878466 0.80 MCHR1 (0.54) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL6878460 0.80 MCHR1 (0.54) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL6875059 0.80 MCHR1 (0.47) MCHR1ADRA2AHRH1ADRA1AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed