SCHEMBL6882020

SCHEMBL6882020

O=C1NCCCc2c1[nH]c1ccccc21

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.81
MEN1 O00255 3/20 0.81
KMT2A Q03164 3/20 0.81
HPGD P15428 2/20 0.81
HTT P42858 2/20 0.81
CYP1A2 P05177 1/20 0.81
CYP2C19 P33261 1/20 0.81
PRKD1 Q15139 1/20 0.67
HSD17B10 Q99714 1/20 0.63
MAPT P10636 3/20 0.54
ALDH1A1 P00352 3/20 0.54
LMNA P02545 2/20 0.54
TUBB4A P04350 1/20 0.52
TUBB P07437 1/20 0.52
TUBA3C P0DPH7 1/20 0.52
TUBA1B P68363 1/20 0.52
TUBA4A P68366 1/20 0.52
TUBB4B P68371 1/20 0.52
TUBB3 Q13509 1/20 0.52
TUBB2A Q13885 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL797563 0.90 KDM4E (1.00) KDM4EMEN1KMT2AHPGDHTT
SCHEMBL9920629 0.80 PRKD1 (1.00) KDM4EMEN1KMT2AHPGDHTT
SCHEMBL21724805 0.80 PRKD1 (0.71) KDM4EMEN1KMT2AHPGDHTT
SCHEMBL15472018 0.80 KDM4E (0.84) KDM4EMEN1KMT2AHPGDHTT
SCHEMBL9920628 0.80 PRKD1 (0.71) KDM4EMEN1KMT2AHPGDHTT
SCHEMBL15868699 0.80 KDM4E (0.79) KDM4EMEN1KMT2AHPGDHTT
SCHEMBL30897563 0.79 MEN1 (0.69) KDM4EMEN1KMT2AHPGDHTT
SCHEMBL4021839 0.77 HSD17B10 (1.00) KDM4EMEN1KMT2AHPGDHTT
SCHEMBL29666273 0.77 HSD17B10 (1.00) KDM4EMEN1KMT2AHPGDHTT
SCHEMBL5239054 0.77 HSD17B10 (0.93) KDM4EMEN1KMT2AHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004098520-A2 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2004-11-18 WO claimed
US-4088647-A Pyrazino (1,2,3-ab)-β-carboline derivatives and salts thereof and method of preparing same GLUSHKOV ROBERT GEORGIEVICH 1978-05-09 US disclosed