SCHEMBL6883447

SCHEMBL6883447

CC(=O)C#Cc1cccc(-c2c(-c3cccs3)c(=O)[nH]c3ccccc23)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 7/20 0.54
MMP2 P08253 4/20 0.38
MMP9 P14780 3/20 0.38
MMP8 P22894 3/20 0.38
MMP13 P45452 3/20 0.38
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
MAPT P10636 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
PPARG P37231 1/20 0.37
KMT2A Q03164 1/20 0.37
NCOA2 Q15596 1/20 0.37
NCOA1 Q15788 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37
PADI4 Q9UM07 1/20 0.36
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL936454 0.87 PDE2A (0.60) PDE2AMMP2MMP9MMP8MMP13
SCHEMBL2681247 0.85 PDE2A (0.54) PDE2AMMP2MMP9MMP8MMP13
SCHEMBL959945 0.85 PDE2A (0.55) PDE2AMMP2MMP9MMP8MMP13
SCHEMBL935286 0.83 PDE2A (0.54) PDE2AMMP2MMP9MMP8MMP13
SCHEMBL936491 0.80 PDE2A (0.54) PDE2AMMP2MMP9MMP8MMP13
SCHEMBL957899 0.79 PDE2A (0.53) PDE2AMMP2MMP9MMP8MMP13
SCHEMBL6352137 0.77 PDE2A (0.48) PDE2AMMP2MMP9MMP8MMP13
SCHEMBL6351761 0.77 PDE2A (0.49) PDE2AMMP2MMP9MMP8MMP13
SCHEMBL958299 0.77 PDE2A (0.49) PDE2AMMP2MMP9MMP8MMP13
SCHEMBL959220 0.77 PDE2A (0.49) PDE2AMMP2MMP9MMP8MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011011312-A1 QUINOLINONE PDE2 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-01-27 WO disclosed