SCHEMBL688385

SCHEMBL688385

CCc1cccc([C@H](CC(=O)O)NC(=O)Nc2c(O)ccn(Cc3ccccc3Cl)c2=O)c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGER3 P43115 17/20 0.51
CYP1A2 P05177 1/20 0.51
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27762474 0.92 PTGER3 (0.42) PTGER3CYP1A2KDM4EALDH1A1MAPK1
SCHEMBL688366 0.91 PTGER3 (0.46) PTGER3CYP1A2KDM4EALDH1A1MAPK1
SCHEMBL687771 0.90 PTGER3 (0.45) PTGER3CYP1A2KDM4EALDH1A1MAPK1
SCHEMBL687732 0.90 PTGER3 (0.49) PTGER3CYP1A2KDM4EALDH1A1MAPK1
SCHEMBL687152 0.90 PTGER3 (0.48) PTGER3CYP1A2KDM4EALDH1A1MAPK1
SCHEMBL687418 0.90 PTGER3 (0.46) PTGER3CYP1A2KDM4EALDH1A1MAPK1
SCHEMBL687654 0.89 PTGER3 (0.43) PTGER3CYP1A2KDM4EALDH1A1MAPK1
SCHEMBL687117 0.89 PTGER3 (0.52) PTGER3CYP1A2KDM4EALDH1A1SMN1; SMN2
SCHEMBL686873 0.88 PTGER3 (0.49) PTGER3CYP1A2KDM4EALDH1A1MAPK1
SCHEMBL687597 0.88 PTGER3 (0.46) PTGER3CYP1A2KDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed