SCHEMBL6884873

SCHEMBL6884873

OC1CCC(Oc2ncc(-c3ccccc3)cn2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
NFKB1 P19838 2/20 0.40
NFKB2 Q00653 2/20 0.40
RELA Q04206 2/20 0.40
PIM1 P11309 1/20 0.39
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
ADORA1 P30542 4/20 0.36
ADORA2A P29274 3/20 0.36
ADORA2B P29275 1/20 0.36
HMOX1 P09601 1/20 0.36
ACACB O00763 3/20 0.36
AKT1 P31749 1/20 0.34
AKT2 P31751 1/20 0.34
HRH1 P35367 1/20 0.34
EPHX2 P34913 1/20 0.34
HTR2B P41595 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6886365 1.00 NPC1 (0.40) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL17698440 0.80 ACACB (0.46) ACACB
SCHEMBL1642513 0.80 ACACB (0.46) ACACB
SCHEMBL1642516 0.80 ACACB (0.46) ACACB
Hydrochloric Acid SCHEMBL2775494 0.79 HRH1 (0.54) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL21192324 0.78 GSK3B (0.36) PIM1ACACB
SCHEMBL718087 0.78 GSK3B (0.36) PIM1ACACB
SCHEMBL16039453 0.77 EPHX2 (0.39) PIM1EPHX2
SCHEMBL16039942 0.77 EPHX2 (0.39) PIM1EPHX2
SCHEMBL719101 0.77 EPHX2 (0.39) PIM1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8389536-B2 Positive allosteric modulators (PAM) HOFFMANN-LA ROCHE INC. (US) 2013-03-05 US disclosed
US-20110098313-A1 POSITIVE ALLOSTERIC MODULATORS (PAM) HOFFMANN-LA ROCHE, INC. 2011-04-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110098313-A1 POSITIVE ALLOSTERIC MODULATORS (PAM) GRM5, GRM1, GRM2 NPC1 3414/4885RAB9A 2271/4885SMN1; SMN2 3467/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.