SCHEMBL6884883

SCHEMBL6884883

O=c1[nH]c2ccc(C=Cc3cccnc3)cc2c(OCC2CCNCC2)c1-c1cccs1

nearest known ligand 0.73

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 8/20 0.73
PADI4 Q9UM07 8/20 0.35
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2681714 0.86 PDE2A (0.76) PDE2AHDAC3HDAC1HDAC2
SCHEMBL2679711 0.84 PDE2A (1.00) PDE2AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL2680306 0.82 PDE2A (0.70) PDE2AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL2680699 0.81 PDE2A (0.68) PDE2AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL2680452 0.80 PDE2A (0.76) PDE2AHDAC3HDAC1HDAC2
SCHEMBL937313 0.79 PDE2A (0.64) PDE2AHDAC3HDAC1HDAC2
SCHEMBL965152 0.79 PDE2A (0.65) PDE2AHDAC3HDAC1HDAC2
SCHEMBL2681127 0.79 PDE2A (0.65) PDE2AHDAC3HDAC1HDAC2
SCHEMBL2680305 0.77 PDE2A (0.63) PDE2AHDAC3HDAC1HDAC2
SCHEMBL2680466 0.77 PDE2A (0.82) PDE2AHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011011312-A1 QUINOLINONE PDE2 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-01-27 WO disclosed