SCHEMBL6886431

SCHEMBL6886431

O=Cc1ccc(OCc2cccc(-c3ccc(Cl)c(C(=O)O)c3)c2)cc1SNC1CC1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.51
ADRA1A P35348 1/20 0.51
HRH1 P35367 1/20 0.51
CYP1A2 P05177 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL804241 0.73 MRGPRX4 (0.60) CYP2C9ADRA1AHRH1CYP1A2
SCHEMBL787619 0.72 CYP2C9 (0.52) CYP2C9ADRA1AHRH1CYP1A2
SCHEMBL804297 0.70 CYP2C9 (0.74) CYP2C9ADRA1AHRH1CYP1A2
SCHEMBL787513 0.69 CYP2C9 (0.97) CYP2C9ADRA1AHRH1
SCHEMBL787603 0.69 CYP2C9 (0.93) CYP2C9ADRA1AHRH1
SCHEMBL787378 0.69 CYP2C9 (0.97) CYP2C9ADRA1AHRH1CYP1A2
SCHEMBL6888905 0.69 MRGPRX4 (0.61) CYP2C9ADRA1AHRH1CYP1A2
SCHEMBL31312330 0.69 CYP2C9 (0.63) CYP2C9ADRA1AHRH1CYP1A2
SCHEMBL787213 0.68 CYP2C9 (0.93) CYP2C9ADRA1AHRH1CYP1A2
SCHEMBL31312311 0.68 CYP2C9 (0.82) CYP2C9ADRA1AHRH1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011116356-A2 POSITIVE ALLOSTERIC MODULATORS OF GROUP II MGLURS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2011-09-22 WO disclosed