SCHEMBL6888093

SCHEMBL6888093

CCc1c(-c2cc[c]cc2)nn(-c2ccccc2C(F)(F)F)c1-c1ccc(O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.44
MAPT P10636 2/20 0.44
MAPK1 P28482 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44
GMNN O75496 1/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
ALOX12 P18054 1/20 0.44
NFKB1 P19838 1/20 0.44
CYP2C19 P33261 1/20 0.44
THPO P40225 1/20 0.44
BLM P54132 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5216937 0.94 ESR1 (0.49) ESR1MAPTMAPK1KMT2AKDM4E
SCHEMBL5222735 0.91 ESR1 (0.47) ESR1MAPTMAPK1KMT2AKDM4E
SCHEMBL5213605 0.87 MAPT (0.43) ESR1MAPTMAPK1KMT2AKDM4E
SCHEMBL5217964 0.87 MAPT (0.43) ESR1MAPTMAPK1KMT2AKDM4E
SCHEMBL5217577 0.85 ESR1 (0.41) ESR1MAPTMAPK1KMT2AKDM4E
SCHEMBL5215618 0.84 ESR1 (0.40) ESR1MAPTMAPK1KMT2AKDM4E
SCHEMBL5217155 0.84 ESR1 (0.40) ESR1MAPTMAPK1KMT2AKDM4E
SCHEMBL5216038 0.83 ESR1 (0.40) ESR1MAPTMAPK1KMT2AKDM4E
SCHEMBL5218923 0.83 ESR1 (0.40) ESR1MAPTMAPK1KMT2AKDM4E
SCHEMBL5214143 0.82 ESR1 (0.40) ESR1MAPTMAPK1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6727273-B2 THERAPY FOR OSTEOPOROSIS, ANTICANCER AGENTS CHIRON CORPORATION 2004-04-27 US disclosed
EP-1102753-A2 PYRAZOLES AS ESTROGEN RECEPTOR MODULATORS CHIRON CORPORATION (US) 2001-05-30 EP disclosed
WO-2000007996-A2 PYRAZOLES AS ESTROGEN RECEPTOR MODULATORS CHIRON CORPORATION (US) 2000-02-17 WO disclosed