SCHEMBL6890622

SCHEMBL6890622

CCOC(=O)CCCC(N)=S

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.61
SMYD3 Q9H7B4 1/20 0.45
GAA P10253 3/20 0.44
ALOX15 P16050 2/20 0.44
MGAM O43451 1/20 0.44
SI P14410 1/20 0.44
MGAM2 Q2M2H8 1/20 0.44
NR1I2 O75469 1/20 0.44
PGR P06401 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
PTGS2 P35354 1/20 0.44
PDE4D Q08499 1/20 0.44
RAB9A P51151 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TDP1 Q9NUW8 2/20 0.43
MAPK1 P28482 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALDH1A1 P00352 2/20 0.42
TSHR P16473 2/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6894888 0.87 CYP1A2 (0.54) CYP1A2GAAALOX15MGAMSI
SCHEMBL11076396 0.85 CYP1A2 (0.68) CYP1A2SMYD3GAAALOX15MGAM
SCHEMBL50734 0.84 CYP1A2 (0.73) CYP1A2SMYD3GAAALOX15MGAM
SCHEMBL1331978 0.84 CYP1A2 (0.73) CYP1A2SMYD3GAAALOX15MGAM
SCHEMBL31150447 0.82 CYP1A2 (0.70) CYP1A2SMYD3GAAALOX15MGAM
Succinic Acid Diethyl Ester SCHEMBL21518140 0.82 CYP1A2 (0.70) CYP1A2SMYD3GAAALOX15MGAM
SCHEMBL8503861 0.81 CYP1A2 (0.57) CYP1A2SMYD3GAAALOX15MGAM
SCHEMBL9509224 0.81 CYP1A2 (0.57) CYP1A2SMYD3GAAALOX15MGAM
SCHEMBL11871882 0.81 CYP1A2 (0.57) CYP1A2SMYD3GAAALOX15MGAM
SCHEMBL11305128 0.80 CYP1A2 (0.68) CYP1A2SMYD3GAAALOX15MGAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP disclosed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP disclosed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO disclosed