SCHEMBL689626

SCHEMBL689626

COc1c(NC(=O)Oc2cc3cccc(CN4CCNCC4)c3n2C)cc(CC(C)C)cc1NS(C)(=O)=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 6/20 0.35
GSK3A P49840 2/20 0.33
ABL1 P00519 1/20 0.32
EGFR P00533 1/20 0.32
RAF1 P04049 1/20 0.32
LYN P07948 1/20 0.32
BRAF P15056 1/20 0.32
EPHA2 P29317 1/20 0.32
EPHA3 P29320 1/20 0.32
AKT1 P31749 1/20 0.32
MAPK9 P45984 1/20 0.32
SCARB1 Q8WTV0 3/20 0.32
MCHR1 Q99705 1/20 0.31
CYP1A2 P05177 1/20 0.31
CHRM2 P08172 1/20 0.31
SLC6A4 P31645 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
CHRM3 P20309 1/20 0.31
MTNR1A P48039 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1303496 0.89 MAPK14 (0.37) MAPK14GSK3AABL1EGFRRAF1
Hydrochloric Acid SCHEMBL688623 0.88 MAPK14 (0.47) MAPK14GSK3AABL1EGFRRAF1
SCHEMBL690048 0.86 MAPK14 (0.46) MAPK14GSK3AABL1EGFRRAF1
SCHEMBL690054 0.85 EPHX2 (0.34) MAPK14ABL1EGFRRAF1LYN
SCHEMBL691275 0.83 MAPK14 (0.40) MAPK14LYNMAPK9SCARB1
SCHEMBL689929 0.83 MAPK14 (0.43) MAPK14GSK3AABL1EGFRRAF1
SCHEMBL689667 0.77 MAPK14 (0.43) MAPK14ABL1EGFRRAF1LYN
SCHEMBL1303413 0.77 MAPK14 (0.49) MAPK14GSK3AABL1EGFRRAF1
SCHEMBL688989 0.77 MAPK14 (0.42) MAPK14ABL1EGFRRAF1LYN
SCHEMBL689461 0.77 DHODH (0.35) MAPK14ABL1EGFRRAF1LYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323980-B1 7-(PIPERAZINE-1-YMETHYL)-1H-INDOLE-2-CARBOXYLIC ACID (PHENYL)-AMIDE DERIVATIVES AND ALLIED COMPOUNDS AS P38 MAP KINASE INHIBITORS FOR THE TREATMENT OF RESPIRATORY DISEASES BOEHRINGER INGELHEIM INT (DE) 2012-02-29 EP disclosed