SCHEMBL6900337

SCHEMBL6900337

CCOc1cn(-c2ccccc2)c(CO)cc1=O

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
COMT P21964 6/20 0.62
GLA P06280 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ELANE P08246 5/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
FGFR1 P11362 1/20 0.38
SRC P12931 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8136252 0.85 COMT (0.56) COMTFGFR1
SCHEMBL14827207 0.80 COMT (0.71) COMT
SCHEMBL6900184 0.79 COMT (0.63) COMT
SCHEMBL1158214 0.78 COMT (0.56) COMTELANEFGFR1SRC
SCHEMBL1157996 0.77 COMT (1.00) COMT
SCHEMBL2434599 0.76 COMT (0.66) COMTSRC
SCHEMBL8138025 0.75 COMT (0.47) COMT
SCHEMBL2467889 0.75 COMT (0.49) COMT
SCHEMBL8136432 0.72 PTPN11 (0.41) COMTFGFR1
SCHEMBL28501968 0.71 COMT (0.45) COMTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011109254-A1 INHIBITORS OF CATECHOL O-METHYL TRANSFERASE AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS MERCK SHARP & DOHME CORP. (US) 2011-09-09 WO disclosed