SCHEMBL6900591

SCHEMBL6900591

CC(C)c1cc(=O)c(O)cn1-c1cccc(-c2ccc3[nH]ccc3c2)c1

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
COMT P21964 9/20 0.69
NPC1 O15118 1/20 0.45
PTGS2 P35354 1/20 0.45
CTSK P43235 3/20 0.43
CTSS P25774 1/20 0.43
GLO1 Q04760 1/20 0.42
MET P08581 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6901910 0.87 COMT (0.67) COMTNPC1
SCHEMBL6901816 0.83 COMT (1.00) COMT
SCHEMBL6901286 0.82 COMT (0.65) COMT
SCHEMBL14816339 0.79 COMT (0.69) COMT
SCHEMBL6900191 0.77 COMT (0.65) COMT
SCHEMBL6901891 0.77 COMT (0.65) COMT
SCHEMBL6900953 0.76 COMT (0.76) COMT
SCHEMBL14816287 0.76 COMT (0.66) COMT
SCHEMBL6899817 0.75 COMT (0.71) COMT
SCHEMBL2439128 0.74 COMT (1.00) COMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011109254-A1 INHIBITORS OF CATECHOL O-METHYL TRANSFERASE AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS MERCK SHARP & DOHME CORP. (US) 2011-09-09 WO disclosed