SCHEMBL6901006

SCHEMBL6901006

CCCSc1ccc2c(C(=O)C(=O)N3CCN(C(=O)c4ccccc4)C[C@H]3C)c[nH]c2n1

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 5/20 0.66
CYP2D6 P10635 4/20 0.66
CYP2C9 P11712 3/20 0.66
CYP3A4 P08684 1/20 0.58
GHSR Q92847 5/20 0.40
SMYD3 Q9H7B4 1/20 0.39
HTT P42858 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SMO Q99835 3/20 0.36
PARP1 P09874 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6431973 0.87 CYP2C19 (0.76) CYP2C19CYP2D6CYP2C9CYP3A4GHSR
SCHEMBL1763412 0.84 CYP2C19 (0.75) CYP2C19CYP2D6CYP2C9CYP3A4GHSR
SCHEMBL1763409 0.84 CYP2C19 (0.75) CYP2C19CYP2D6CYP2C9CYP3A4GHSR
SCHEMBL6431861 0.84 CYP2C19 (0.74) CYP2C19CYP2D6CYP2C9CYP3A4GHSR
SCHEMBL1763475 0.83 CYP2C19 (0.73) CYP2C19CYP2D6CYP2C9CYP3A4GHSR
SCHEMBL1763473 0.83 CYP2C19 (0.73) CYP2C19CYP2D6CYP2C9CYP3A4GHSR
SCHEMBL6435656 0.83 CYP2C19 (0.67) CYP2C19CYP2D6CYP2C9CYP3A4GHSR
SCHEMBL1763438 0.81 CYP2C19 (0.70) CYP2C19CYP2D6CYP2C9CYP3A4GHSR
SCHEMBL1763436 0.81 CYP2C19 (0.70) CYP2C19CYP2D6CYP2C9CYP3A4GHSR
SCHEMBL6435698 0.81 CYP2D6 (0.70) CYP2C19CYP2D6CYP2C9CYP3A4GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1257276-A4 ANTIVIRAL AZAINDOLE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2004-10-27 EP disclosed
EP-1257276-A1 ANTIVIRAL AZAINDOLE DERIVATIVES BRISTOL-MYERS SQUIBB COMPANY (US) 2002-11-20 EP disclosed
WO-2001062255-A1 ANTIVIRAL AZAINDOLE DERIVATIVES BRISTOL-MYERS SQUIBB COMPANY (US) 2001-08-30 WO disclosed