SCHEMBL6901025

SCHEMBL6901025

Cc1cccc(-c2cccc(-n3cc(O)c(=O)cc3C(C)O)c2)c1

nearest known ligand 0.83

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
COMT P21964 12/20 0.83
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2439128 0.91 COMT (1.00) COMT
SCHEMBL14815720 0.86 COMT (0.81) COMT
SCHEMBL6901028 0.85 COMT (0.84) COMT
SCHEMBL6901182 0.83 COMT (0.76) COMT
SCHEMBL6900331 0.83 COMT (0.76) COMT
SCHEMBL22878777 0.83 COMT (0.67) COMT
SCHEMBL6901158 0.82 COMT (0.74) COMT
SCHEMBL6901163 0.82 COMT (0.74) COMT
SCHEMBL6901816 0.82 COMT (1.00) COMT
SCHEMBL14816342 0.82 COMT (0.73) COMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011109254-A1 INHIBITORS OF CATECHOL O-METHYL TRANSFERASE AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS MERCK SHARP & DOHME CORP. (US) 2011-09-09 WO disclosed