SCHEMBL6901998

SCHEMBL6901998

Cc1cc(-c2cccc(-n3cc(O)c(=O)cc3C)c2)ccn1

nearest known ligand 0.72

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
COMT P21964 9/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14827143 0.86 COMT (0.66) COMT
SCHEMBL2465251 0.84 COMT (1.00) COMT
SCHEMBL6900252 0.77 COMT (0.64) COMT
SCHEMBL6900999 0.77 COMT (0.63) COMT
SCHEMBL14827138 0.77 COMT (0.60) COMT
SCHEMBL23249865 0.75 DYRK1A (0.44) COMT
SCHEMBL6901910 0.75 COMT (0.67) COMT
SCHEMBL6900222 0.75 COMT (0.64) COMT
SCHEMBL14827201 0.75 COMT (0.77) COMT
SCHEMBL19331190 0.73 COMT (0.66) COMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011109254-A1 INHIBITORS OF CATECHOL O-METHYL TRANSFERASE AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS MERCK SHARP & DOHME CORP. (US) 2011-09-09 WO disclosed