SCHEMBL690221

SCHEMBL690221

COc1c(CN2CCN(C)CC2)cc(C(C)(C)C)cc1NC(=O)Oc1cc2cccc(CN3CCN(C(=O)[C@@H]4CCCN4C)CC3)c2n1C

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 3/20 0.36
SSTR5 P35346 1/20 0.36
EPHX2 P34913 1/20 0.35
DHODH Q02127 2/20 0.33
GSK3A P49840 2/20 0.33
LYN P07948 1/20 0.32
MAPK9 P45984 1/20 0.32
KDM4E B2RXH2 2/20 0.32
TSHR P16473 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK14 Q16539 3/20 0.32
BRAF P15056 1/20 0.32
RORC P51449 1/20 0.32
FAAH O00519 1/20 0.31
RET P07949 1/20 0.31
CHRM3 P20309 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688611 0.95 ACKR3 (0.37) ACKR3SSTR5EPHX2DHODHGSK3A
SCHEMBL690441 0.94 ACKR3 (0.35) ACKR3SSTR5EPHX2DHODHLYN
SCHEMBL689257 0.93 ACKR3 (0.36) ACKR3SSTR5EPHX2DHODHLYN
SCHEMBL690851 0.93 EPHX2 (0.35) ACKR3SSTR5EPHX2DHODHLYN
SCHEMBL690908 0.92 ACKR3 (0.35) ACKR3SSTR5EPHX2DHODHLYN
SCHEMBL690495 0.92 ACKR3 (0.34) ACKR3SSTR5EPHX2DHODHGSK3A
SCHEMBL689757 0.92 ACKR3 (0.35) ACKR3SSTR5EPHX2DHODHGSK3A
SCHEMBL689851 0.92 EPHX2 (0.35) ACKR3SSTR5EPHX2DHODHGSK3A
SCHEMBL690660 0.92 ACKR3 (0.34) ACKR3SSTR5EPHX2DHODHGSK3A
SCHEMBL689541 0.92 EPHX2 (0.36) ACKR3SSTR5EPHX2DHODHGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323980-B1 7-(PIPERAZINE-1-YMETHYL)-1H-INDOLE-2-CARBOXYLIC ACID (PHENYL)-AMIDE DERIVATIVES AND ALLIED COMPOUNDS AS P38 MAP KINASE INHIBITORS FOR THE TREATMENT OF RESPIRATORY DISEASES BOEHRINGER INGELHEIM INT (DE) 2012-02-29 EP claimed
EP-2323980-B1 7-(PIPERAZINE-1-YMETHYL)-1H-INDOLE-2-CARBOXYLIC ACID (PHENYL)-AMIDE DERIVATIVES AND ALLIED COMPOUNDS AS P38 MAP KINASE INHIBITORS FOR THE TREATMENT OF RESPIRATORY DISEASES BOEHRINGER INGELHEIM INT (DE) 2012-02-29 EP disclosed