SCHEMBL690414

SCHEMBL690414

N#Cc1ccccc1-c1ccc(C=CC(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 4/20 0.54
HDAC2 Q92769 3/20 0.53
HCAR2 Q8TDS4 2/20 0.53
HDAC3 O15379 1/20 0.53
TNKS O95271 1/20 0.53
HDAC4 P56524 1/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53
HDAC10 Q969S8 1/20 0.53
HDAC11 Q96DB2 1/20 0.53
HDAC8 Q9BY41 1/20 0.53
TNKS2 Q9H2K2 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
HDAC9 Q9UKV0 1/20 0.53
HDAC5 Q9UQL6 1/20 0.53
FFAR1 O14842 3/20 0.51
SLC22A12 Q96S37 1/20 0.47
PTPN5 P54829 1/20 0.47
ALDH1A1 P00352 2/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873052 0.84 HDAC1 (0.49) ESR2HDAC2HCAR2HDAC3TNKS
SCHEMBL31325636 0.79 ESR2 (0.42) ESR2HDAC2HCAR2HDAC3TNKS
SCHEMBL526946 0.78 CA1 (0.50) ESR2HDAC2HCAR2HDAC3TNKS
SCHEMBL8641083 0.78 HDAC2 (0.60) ESR2HDAC2HCAR2HDAC3TNKS
SCHEMBL28887390 0.78 BACE1 (0.64) ESR2HDAC2HCAR2HDAC3TNKS
SCHEMBL29576664 0.78 BACE1 (0.64) ESR2HDAC2HCAR2HDAC3TNKS
SCHEMBL8973589 0.78 HDAC2 (0.60) ESR2HDAC2HCAR2HDAC3TNKS
Acrylic Acid SCHEMBL211815 0.78 ESR2 (0.56) ESR2FFAR1PTPN5ALDH1A1L3MBTL1
SCHEMBL2572 0.77 ESR2 (0.59) ESR2FFAR1PTPN5ALDH1A1AKR1B1
Cinnamic Acid SCHEMBL29454354 0.77 HDAC2 (0.76) ESR2HDAC2HCAR2HDAC3TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0982356-A2 Improved stabilized coatings Clariant Finance (BVI) Limited (VG) 2000-03-01 EP claimed
EP-4051216-A1 POLYSACCHARIDE-BASED GELLED FOAM URGO RECHERCHE INNOVATION ET DEVELOPPEMENT (FR) 2022-09-07 EP disclosed
WO-2021084200-A1 POLYSACCHARIDE-BASED GELLED FOAM URGO RECHERCHE INNOVATION ET DEVELOPPEMENT (FR) 2021-05-06 WO disclosed
EP-3544573-A1 FILM-FORMING COMPOSITION Urgo Recherche Innovation et Développement (FR) 2019-10-02 EP disclosed
EP-3125859-B1 FILM-FORMING COMPOSITION URGO RECH INNOVATION ET DEVELOPPEMENT (FR) 2019-06-12 EP disclosed
EP-2968197-B1 FILM-FORMING COMPOSITION AND USE THEREOF FOR THE TREATMENT OF SKIN DISORDERS URGO RECH INNOVATION ET DEVELOPPEMENT (FR) 2018-12-26 EP disclosed
WO-2018178597-A1 COMPOSITION CONTAINING A CELLULOSE DERIVATIVE, A PLASTICISER AND A VOLATILE SOLVENT, AND ITS USES AS A DRESSING URGO RECHERCHE INNOVATION ET DEVELOPPEMENT (FR) 2018-10-04 WO disclosed
WO-2018096224-A1 FILM-FORMING COMPOSITION URGO RECHERCHE INNOVATION ET DEVELOPPEMENT (FR) 2018-05-31 WO disclosed
EP-3125859-A1 FILM-FORMING COMPOSITION Laboratoires Urgo (FR) 2017-02-08 EP disclosed
EP-2688651-B1 COMPOSITION COTAINING A CELLULOSE, A VEGETAL OIL AND A VOLATILE SOLVENT, ITS USE AS WOUND DRESSING URGO RECH INNOVATION ET DEVELOPPEMENT (FR) 2016-12-28 EP disclosed
EP-2861201-A1 AQUEOUS DISPERSION OF POLYMER PARTICLES, FILM-FORMING COMPOSITION CONTAINING SAME AND USES THEREOF Vivatech (FR) 2015-04-22 EP disclosed
EP-2793946-A1 TOPICAL FILM-FORMING COMPOSITION, AND USE THEREOF FOR TREATING OR PREVENTING ONYCHOPHAGIA Laboratoires Urgo (FR) 2014-10-29 EP disclosed
WO-2014140475-A1 FILM-FORMING COMPOSITION AND USE THEREOF FOR THE TREATMENT OF SKIN DISORDERS LABORATOIRES URGO (FR) 2014-09-18 WO disclosed
EP-2688651-A1 COMPOSITION CONTAINING A CELLULOSE, A VEGETABLE OIL AND A VOLATILE SOLVENT, AND USE THEREOF AS A DRESSING Laboratoires Urgo (FR) 2014-01-29 EP disclosed
WO-2013182828-A1 AQUEOUS DISPERSION OF POLYMER PARTICLES, FILM-FORMING COMPOSITION CONTAINING SAME AND USES THEREOF SOCIETE DE DEVELOPPEMENT ET DE RECHERCHE INDUSTRIELLE (FR) 2013-12-12 WO disclosed
WO-2013093216-A1 TOPICAL FILM-FORMING COMPOSITION, AND USE THEREOF FOR TREATING OR PREVENTING ONYCHOPHAGIA LABORATOIRES URGO (FR) 2013-06-27 WO disclosed
WO-2012131238-A1 COMPOSITION CONTAINING A CELLULOSE, A VEGETABLE OIL AND A VOLATILE SOLVENT, AND USE THEREOF AS A DRESSING LABORATOIRES URGO (FR) 2012-10-04 WO disclosed
EP-2421495-A2 METHOD FOR FORMING CYCLODEXTRIN POLYMER AND LIPOPHILIC COMPOUND EMULSIONS, RESULTING EMULSIONS, AND COMPOSITIONS INCLUDING SAID EMULSIONS Centre National De La Recherche Scientifique CNRS (FR) 2012-02-29 EP disclosed
WO-2010122246-A2 METHOD FOR FORMING CYCLODEXTRIN POLYMER AND LIPOPHILIC COMPOUND EMULSIONS, RESULTING EMULSIONS, AND COMPOSITIONS INCLUDING SAID EMULSIONS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE -CNRS - (FR) 2010-10-28 WO disclosed
EP-0982356-A2 Improved stabilized coatings Clariant Finance (BVI) Limited (VG) 2000-03-01 EP disclosed