SCHEMBL6911478

SCHEMBL6911478

CCOC(=O)/C=C/c1ccc(F)cc1C(C#N)(CC)CC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.43
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
TTR P02766 1/20 0.40
DPP4 P27487 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
EPAS1 Q99814 1/20 0.40
CYP3A4 P08684 2/20 0.39
MAPT P10636 4/20 0.39
POLB P06746 1/20 0.39
RAB9A P51151 1/20 0.39
HSD17B1 P14061 1/20 0.38
HSD17B2 P37059 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1508785 0.84 ESR1 (0.47) ESR1IDO1TDO2TTRDPP4
SCHEMBL1508701 0.84 ESR1 (0.47) ESR1IDO1TDO2TTRDPP4
SCHEMBL11353373 0.80 TTR (0.44) ESR1IDO1TDO2TTRDPP4
SCHEMBL11353377 0.80 TTR (0.44) ESR1IDO1TDO2TTRDPP4
SCHEMBL23201588 0.80 TTR (0.46) ESR1IDO1TDO2TTRDPP4
SCHEMBL4514544 0.78 ESR1 (0.57) ESR1IDO1TDO2TTRDPP4
SCHEMBL8375820 0.78 POLB (0.56) ESR1IDO1TDO2TTRDPP4
SCHEMBL30235603 0.78 ESR1 (0.57) ESR1IDO1TDO2TTRDPP4
SCHEMBL8375818 0.78 POLB (0.56) ESR1IDO1TDO2TTRDPP4
SCHEMBL13678677 0.78 ESR1 (0.57) ESR1IDO1TDO2TTRDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046771-A1 SUBSTITUTED PIPERIDINES THAT INCREASE p53 ACTIVITY AND THE USES THEREOF SCHERING CORPORATION (US) 2011-04-21 WO disclosed