SCHEMBL6915733

SCHEMBL6915733

O=S(=O)(Cc1ccccc1Cl)c1ccc2[nH]c(-c3cccc(Cl)n3)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 10/20 0.46
CYP1A2 P05177 10/20 0.46
CYP3A4 P08684 10/20 0.46
CYP2C19 P33261 9/20 0.46
CYP2D6 P10635 5/20 0.46
CBFB Q13951 2/20 0.39
KDM4E B2RXH2 1/20 0.38
KMT2A Q03164 1/20 0.38
EGLN1 Q9GZT9 1/20 0.38
GRM4 Q14833 1/20 0.38
AKR1B1 P15121 1/20 0.37
SCD O00767 1/20 0.37
OPRL1 P41146 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12689566 0.90 CYP2C9 (0.47) CYP2C9CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL6915839 0.90 CYP1A2 (0.44) CYP2C9CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL1822351 0.87 CBFB (0.55) CYP2C9CYP1A2CYP3A4CYP2C19CBFB
SCHEMBL6916201 0.82 METAP1 (0.51) CYP2C9CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL6915845 0.81 CBFB (0.50) CYP2C9CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL6925674 0.80 MAPT (0.49) KDM4EKMT2AGRM4
SCHEMBL6915491 0.78 CBFB (0.54) CYP2C9CYP1A2CYP3A4CYP2C19CBFB
SCHEMBL12689481 0.78 GRM4 (0.42) CYP2C9CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL12689474 0.78 EGLN1 (0.38) CYP2C9CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL6915101 0.78 CBFB (0.41) CYP2C9CYP1A2CYP3A4CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011057208-A2 ARYL AND HETEROARYL SULFONES AS MGLUR4 ALLOSTERIC POTENTIATORS, COMPOSITIONS, AND METHODS OF TREATING NEUROLOGICAL DYSFUNCTION VANDERBILT UNIVERSITY (US) 2011-05-12 WO disclosed