Niludipine

Niludipine

SCHEMBL691639

CCCOCCOC(=O)C1=C(C)NC(C)=C(C(=O)OCCOCCC)C1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.84

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1F O60840 9/20 0.84
CACNA1D Q01668 9/20 0.84
CACNA1S Q13698 9/20 0.84
CACNA1C Q13936 9/20 0.84
ADORA3 P0DMS8 1/20 0.78
MEN1 O00255 4/20 0.72
CYP1A2 P05177 4/20 0.72
CYP3A4 P08684 4/20 0.72
CYP2C9 P11712 4/20 0.72
CYP2C19 P33261 4/20 0.72
KMT2A Q03164 4/20 0.72
HIF1A Q16665 3/20 0.72
MAPT P10636 3/20 0.72
LMNA P02545 3/20 0.72
CYP2D6 P10635 2/20 0.72
TSHR P16473 2/20 0.72
NFKB1 P19838 2/20 0.72
THPO P40225 2/20 0.72
POLB P06746 1/20 0.72
MAPK1 P28482 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11829739 0.98 CACNA1F (0.88) CACNA1FCACNA1DCACNA1SCACNA1CADORA3
SCHEMBL11839673 0.96 MEN1 (0.80) CACNA1FCACNA1DCACNA1SCACNA1CADORA3
SCHEMBL9765729 0.96 CACNA1C (0.78) CACNA1FCACNA1DCACNA1SCACNA1CADORA3
SCHEMBL7282379 0.95 CACNA1F (0.76) CACNA1FCACNA1DCACNA1SCACNA1CADORA3
SCHEMBL9765763 0.94 MEN1 (0.82) CACNA1FCACNA1DCACNA1SCACNA1CADORA3
SCHEMBL11005401 0.94 CACNA1F (0.74) CACNA1FCACNA1DCACNA1SCACNA1CADORA3
SCHEMBL6725228 0.94 CACNA1F (0.87) CACNA1FCACNA1DCACNA1SCACNA1CADORA3
SCHEMBL11688627 0.93 CACNA1F (0.90) CACNA1FCACNA1DCACNA1SCACNA1CADORA3
SCHEMBL10989784 0.93 CACNA1C (0.72) CACNA1FCACNA1DCACNA1SCACNA1CADORA3
SCHEMBL7439297 0.92 CACNA1F (0.72) CACNA1FCACNA1DCACNA1SCACNA1CADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 463 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4301370-A1 COMBINATORY THERAPY FOR PREVENTING, INHIBITING, TREATING, OR REDUCING ANEURYSMS The Regents of The University of California (US) 2024-01-10 EP claimed
US-20230330188-A1 PHARMACEUTICAL COMBINATION FOR USE IN THE TREATMENT AND/OR PREVENTION OF DIABETES INSPHERO AG (CH) 2023-10-19 US claimed
EP-4225296-A1 PHARMACEUTICAL COMBINATION FOR USE IN THE TREATMENT AND/OR PREVENTION OF DIABETES Insphero AG (CH) 2023-08-16 EP claimed
EP-3498297-B1 PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF AUTISM STALICLA S A (CH) 2023-06-21 EP claimed
WO-2022187349-A1 COMBINATORY THERAPY FOR PREVENTING, INHIBITING, TREATING, OR REDUCING ANEURYSMS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-09-09 WO claimed
WO-2022074057-A1 PHARMACEUTICAL COMBINATION FOR USE IN THE TREATMENT AND/OR PREVENTION OF DIABETES INSPHERO AG (CH) 2022-04-14 WO claimed
EP-3981401-A1 PHARMACEUTICAL COMBINATION FOR THE TREATMENT AND/OR PREVENTION OF DIABETES COMPRISING A CALCIUM CHANNEL BLOCKING AGENT AND AN INCRETIN MIMETIC InSphero AG (CH) 2022-04-13 EP claimed
EP-2649989-B1 Method for preparing a solid dispersion, solid dispersion obtained thereby and use thereof UNIV KING SAUD (SA) 2017-10-18 EP claimed
EP-2575473-B1 SOLUBLE GUANYLATE CYCLASE ACTIVATORS MERCK SHARP & DOHME (US) 2016-01-20 EP claimed
EP-2649989-A1 Method for preparing a solid dispersion, solid dispersion obtained thereby and use thereof King Saud University (SA) 2013-10-16 EP claimed
EP-0412594-B1 Substituted triazolinones, triazolinethiones, and triazolinimines as angiotensin II antagonists MERCK & CO INC (US) 1996-01-03 EP claimed
EP-0330924-B1 Use of 1,4-dihydropyridine derivatives in the treatment of alcohol addiction TROPONWERKE GMBH & CO KG (DE) 1995-05-24 EP claimed
EP-0411766-B1 Substituted quinazolinones as angiotensin II antagonists MERCK & CO INC (US) 1994-01-19 EP claimed
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP claimed
EP-0319983-B1 ASSOCIATION OF PYRIMIDINE DERIVATIVES AND CALCIUM ANTAGONISTS TO INDUCE AND STIMULATE THE HAIR GROWTH AND TO REDUCE HAIR LOSS L'OREAL (FR) 1992-06-03 EP claimed
EP-0317780-B1 SUSTAINED (CONTROLLED) RELEASE DELIVERY SYSTEM FOR SUBSTITUTED DIHYDROPYRIDINE CALCIUM CHANNEL BLOCKERS AMERICAN CYANAMID COMPANY (US) 1992-05-20 EP claimed
EP-0237506-B1 PHARMACEUTICAL COMPOSITION LEJUS MEDICAL AKTIEBOLAG (SE) 1991-08-14 EP claimed
EP-0293714-B1 COMBINATIONS OF COMPOUNDS WITH ANTI-DEPRESSIVE ACTIVITY Troponwerke GmbH & Co. KG (DE) 1991-06-05 EP claimed
EP-0330924-A2 Use of 1,4-dihydropyridine derivatives in the treatment of alcohol addiction Troponwerke GmbH & Co. KG (DE) 1989-09-06 EP claimed
US-4618598-A Method of regulating hormone function or release DUKE UNIVERSITY (US) 1986-10-21 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230330188-A1 PHARMACEUTICAL COMBINATION FOR USE IN THE TREATMENT AND/OR PREVENTION OF DIABETES IAPP, SLC5A2, GLP1R CACNA1F 11/4885CACNA1D 16/4885CACNA1S 22/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.