SCHEMBL6918671

SCHEMBL6918671

Nc1ccc(NC(=O)c2cc(F)cc(Oc3cncnc3)c2)nc1

nearest known ligand 0.81

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.67
CYP3A4 P08684 3/20 0.67
DRD3 P35462 1/20 0.57
SLC6A3 Q01959 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6918223 0.90 GRM5 (0.81) GRM5CYP3A4
SCHEMBL6918225 0.87 GRM5 (0.77) GRM5CYP3A4
SCHEMBL12602061 0.86 GRM5 (0.66) GRM5CYP3A4
SCHEMBL6919980 0.85 GRM5 (0.76) GRM5CYP3A4
SCHEMBL6918543 0.83 GRM5 (0.73) GRM5CYP3A4
SCHEMBL6918725 0.82 GRM5 (0.82) GRM5CYP3A4
SCHEMBL6918698 0.80 GRM5 (0.77) GRM5CYP3A4
SCHEMBL6918336 0.80 GRM5 (1.00) GRM5CYP3A4
SCHEMBL6918747 0.80 GRM5 (0.66) GRM5CYP3A4DRD3SLC6A3
SCHEMBL6918375 0.79 GRM5 (0.77) GRM5CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011035209-A1 SUBSTITUTED BENZAMIDE ANALOGS AS MGLUR5 NEGATIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING THE SAME VANDERBILT UNIVERSTIY (US) 2011-03-24 WO disclosed