SCHEMBL6918685

SCHEMBL6918685

NC(=O)[C@@H]1C[C@@H](F)CN1Cc1cc(Cl)ccc1-n1cnnn1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 7/20 0.44
MAOB P27338 7/20 0.44
GPBAR1 Q8TDU6 2/20 0.43
CYP3A4 P08684 3/20 0.42
F2 P00734 6/20 0.42
PRSS1 P07477 2/20 0.42
F9 P00740 1/20 0.42
F10 P00742 1/20 0.42
PLAT P00750 1/20 0.42
F11 P03951 1/20 0.42
KLKB1 P03952 1/20 0.42
F7 P08709 1/20 0.42
TBXA2R P21731 1/20 0.42
PRSS3 P35030 1/20 0.42
MASP2 O00187 1/20 0.40
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6919450 0.84 MAOB (0.44) MAOAMAOBGPBAR1F2
SCHEMBL6914971 0.84 MAOB (0.44) MAOAMAOBGPBAR1F2
Hydrochloric Acid SCHEMBL6920555 0.83 MAOB (0.43) MAOAMAOBGPBAR1F2
Hydrochloric Acid SCHEMBL6919805 0.83 MAOB (0.43) MAOAMAOBGPBAR1F2
SCHEMBL6921701 0.82 GPBAR1 (0.45) MAOAMAOBGPBAR1CYP3A4F2
SCHEMBL6922183 0.82 CYP3A4 (0.48) GPBAR1CYP3A4F2PRSS1F9
SCHEMBL6078656 0.82 F2 (0.47) GPBAR1CYP3A4F2PRSS1F9
Hydrochloric Acid SCHEMBL6079141 0.81 F2 (0.46) GPBAR1CYP3A4F2PRSS1F9
SCHEMBL6918997 0.81 CYP3A4 (0.45) GPBAR1CYP3A4F2PRSS1F9
SCHEMBL6916861 0.81 CYP3A4 (0.45) GPBAR1CYP3A4F2PRSS1F9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004032834-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2004-04-22 WO disclosed