SCHEMBL6919488

SCHEMBL6919488

COC(=O)c1cccc2ccn(CCN)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
CFTR P13569 1/20 0.41
USP2 O75604 1/20 0.40
MAPK1 P28482 1/20 0.40
LMNA P02545 3/20 0.38
TSHR P16473 2/20 0.38
KDM4E B2RXH2 4/20 0.38
MAPT P10636 2/20 0.38
TLR8 Q9NR97 1/20 0.37
MAPK8 P45983 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA5A P35218 1/20 0.37
CA9 Q16790 1/20 0.37
KMT2A Q03164 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18394802 0.87 CNR2 (0.44) ALDH1A1HSD17B10CFTRUSP2MAPK1
SCHEMBL29664577 0.87 CNR2 (0.44) ALDH1A1HSD17B10CFTRUSP2MAPK1
SCHEMBL13557127 0.85 MAPK1 (0.44) ALDH1A1HSD17B10CFTRUSP2MAPK1
SCHEMBL1078681 0.84 MAPK1 (0.39) ALDH1A1HSD17B10CFTRUSP2MAPK1
SCHEMBL1080174 0.83 MAPK1 (0.38) ALDH1A1HSD17B10CFTRUSP2MAPK1
SCHEMBL1077377 0.81 NR4A2 (0.39) ALDH1A1HSD17B10CFTRUSP2MAPK1
SCHEMBL12584098 0.80 KDM4E (0.41) ALDH1A1USP2MAPK1TSHRKDM4E
SCHEMBL22800161 0.80 CYP3A4 (0.38) ALDH1A1HSD17B10USP2MAPK1LMNA
SCHEMBL12584050 0.80 KDM4E (0.47) ALDH1A1HSD17B10TSHRKDM4EMAPT
SCHEMBL12750465 0.80 KDM4E (0.43) ALDH1A1HSD17B10CFTRUSP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011008572-A2 5-HT3 RECEPTOR MODULATORS, METHODS OF MAKING, AND USE THEREOF ALBANY MOLECULAR RESEARCH, INC. (US) 2011-01-20 WO disclosed