SCHEMBL6920144

SCHEMBL6920144

O=C(Nc1ccccc1Br)N(c1c(O)c(F)cc(F)c1F)N(C(=O)Nc1ccccc1Br)c1c(O)c(F)cc(F)c1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.50
ALDH1A1 P00352 3/20 0.45
CXCR1 P25024 6/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.41
CXCR2 P25025 6/20 0.41
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TOP1 P11387 1/20 0.39
TOP2A P11388 1/20 0.39
TOP2B Q02880 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5594846 0.78 HTT (0.61) HTTALDH1A1CXCR1NPC1RAB9A
SCHEMBL6920143 0.78 HTT (0.61) HTTALDH1A1CXCR1NPC1RAB9A
SCHEMBL5594969 0.71 HTT (0.65) HTTALDH1A1CXCR1NPC1RAB9A
SCHEMBL5594682 0.70 HTT (0.67) HTTALDH1A1CXCR1NPC1RAB9A
SCHEMBL6825931 0.69 HTT (0.76) HTTALDH1A1CXCR1NPC1RAB9A
SCHEMBL5595083 0.69 HTT (0.76) HTTALDH1A1CXCR1NPC1RAB9A
SCHEMBL4139764 0.69 HTT (0.53) HTTALDH1A1CXCR1NPC1RAB9A
SCHEMBL27517285 0.68 CA1 (0.32) HTTALDH1A1CXCR1NPC1RAB9A
SCHEMBL7488566 0.68 HTT (0.62) HTTALDH1A1CXCR1NPC1RAB9A
SCHEMBL6823585 0.67 CXCR1 (0.55) HTTCXCR1NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1185261-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-02-25 EP disclosed
EP-1185261-A1 IL-8 RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2002-03-13 EP disclosed
WO-2000076495-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2000-12-21 WO disclosed