SCHEMBL6920640

SCHEMBL6920640

NC(=O)c1cc(Cl)cc(Oc2cncnc2)c1

nearest known ligand 0.57

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.55
CYP3A4 P08684 4/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1487645 0.86 GRM5 (0.56) GRM5CYP3A4
SCHEMBL1981351 0.82 GRM5 (0.59) GRM5CYP3A4
SCHEMBL6919814 0.81 GRM5 (0.55) GRM5CYP3A4
SCHEMBL6919417 0.76 GRM5 (0.65) GRM5CYP3A4
SCHEMBL2182610 0.75 GRM5 (0.43) GRM5CYP3A4
SCHEMBL6918719 0.74 CYP3A4 (0.81) GRM5CYP3A4
SCHEMBL7448823 0.73 PARP1 (0.55)
SCHEMBL6918743 0.73 GRM5 (0.62) GRM5CYP3A4
SCHEMBL6919023 0.73 GRM5 (0.82) GRM5CYP3A4
SCHEMBL2180716 0.73 GRM5 (0.52) GRM5CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011035209-A1 SUBSTITUTED BENZAMIDE ANALOGS AS MGLUR5 NEGATIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING THE SAME VANDERBILT UNIVERSTIY (US) 2011-03-24 WO disclosed