SCHEMBL6921764

SCHEMBL6921764

COc1c(C)cc([C@]2(c3cccc(-c4cncnc4)c3)N=C(C)C(N)=N2)cc1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 1.00
BACE2 Q9Y5Z0 3/20 1.00
KCNH2 Q12809 8/20 0.72
REN P00797 1/20 0.48
CTSD P07339 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931641 1.00 BACE1 (1.00) BACE1BACE2KCNH2RENCTSD
SCHEMBL931639 1.00 BACE1 (1.00) BACE1BACE2KCNH2RENCTSD
SCHEMBL932576 0.90 BACE1 (0.82) BACE1BACE2KCNH2RENCTSD
SCHEMBL932133 0.88 BACE1 (0.78) BACE1BACE2KCNH2RENCTSD
SCHEMBL931689 0.88 BACE1 (1.00) BACE1BACE2KCNH2RENCTSD
SCHEMBL932012 0.88 BACE1 (0.78) BACE1BACE2KCNH2
SCHEMBL931679 0.87 BACE1 (0.77) BACE1BACE2KCNH2
SCHEMBL932314 0.86 BACE1 (0.76) BACE1BACE2KCNH2RENCTSD
SCHEMBL932620 0.85 BACE1 (1.00) BACE1BACE2KCNH2CTSD
SCHEMBL931666 0.85 BACE1 (0.74) BACE1BACE2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed