SCHEMBL6921976

SCHEMBL6921976

CN(C)CCOc1ccc(NC(=O)c2ccc(-c3ccccc3)cc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 9/20 0.77
KDR P35968 1/20 0.59
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57
TSHR P16473 1/20 0.57
RAB9A P51151 1/20 0.57
MCL1 Q07820 1/20 0.57
HSD17B10 Q99714 1/20 0.57
HRH3 Q9Y5N1 1/20 0.56
LSS P48449 1/20 0.56
CACNA1H O95180 1/20 0.56
CACNA1B Q00975 1/20 0.56
CHRNB2 P17787 2/20 0.55
CHRNB4 P30926 2/20 0.55
CHRNA3 P32297 2/20 0.55
CHRNA7 P36544 2/20 0.55
CHRNA4 P43681 2/20 0.55
CHRNA10 Q9GZZ6 1/20 0.55
CHRNA9 Q9UGM1 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6924167 0.94 MCHR1 (0.71) MCHR1KDRKDM4EALDH1A1MAPT
SCHEMBL6803781 0.87 MCHR1 (1.00) MCHR1
SCHEMBL6920369 0.87 MCHR1 (0.68) MCHR1MAPTRAB9AMCL1
SCHEMBL6928640 0.82 MCHR1 (0.92) MCHR1KDM4EALDH1A1MAPTHSD17B10
SCHEMBL6928025 0.81 MAOB (0.66) MCHR1KDRKDM4EALDH1A1MAPT
SCHEMBL22831331 0.81 LSS (0.83) KDM4EALDH1A1MAPTRAB9AHRH3
SCHEMBL5582704 0.81 MCHR1 (0.70) MCHR1KDM4EMAPTRAB9APTPN1
SCHEMBL6929529 0.80 MCHR1 (0.65) MCHR1KDM4EALDH1A1CACNA1HCACNA1B
SCHEMBL16712946 0.80 MCHR1 (0.61) MCHR1KDRHRH3
SCHEMBL8126082 0.80 RARB (0.63) KDM4ETSHRLSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6515027-B1 Ligands, agonists or antagonists, of the CC chemokine receptor CC-CKR5 SMITHKLINE BEECHAM CORP. 2003-02-04 US disclosed
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed