SCHEMBL6922543

SCHEMBL6922543

Nc1cncc(Br)c1.O=C(O)c1c2n(c3c(N4CCN(CCc5ccc(F)c(F)c5)CC4)ncnc13)CCCC2

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 20/20 0.72
CYP3A4 P08684 8/20 0.72
ABCG2 Q9UNQ0 2/20 0.46
ABCB1 P08183 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822285 0.90 ABCC1 (0.85) ABCC1CYP3A4ABCG2ABCB1
SCHEMBL6920782 0.84 ABCC1 (1.00) ABCC1CYP3A4
SCHEMBL7172529 0.84 ABCC1 (0.73) ABCC1CYP3A4
SCHEMBL6919449 0.83 ABCC1 (0.98) ABCC1CYP3A4ABCG2
SCHEMBL6919172 0.83 ABCC1 (0.97) ABCC1CYP3A4
SCHEMBL6919932 0.80 ABCC1 (0.86) ABCC1CYP3A4ABCG2ABCB1
SCHEMBL6918024 0.80 ABCC1 (0.85) ABCC1CYP3A4ABCG2ABCB1
SCHEMBL6917967 0.79 ABCC1 (1.00) ABCC1CYP3A4ABCG2ABCB1
SCHEMBL6822752 0.79 ABCC1 (0.68) ABCC1CYP3A4
SCHEMBL6823384 0.79 ABCC1 (0.86) ABCC1CYP3A4ABCG2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004065389-A1 PYRROLOPYRIMIDINE DERIVATIVES USEFUL AS MODULATORS OF MULTIDRUG RESISTANCE XENOVA LIMITED (GB) 2004-08-05 WO claimed