SCHEMBL6922787

SCHEMBL6922787

Nc1cc(Cl)cc(Nc2noc3cccnc23)c1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.55
GRM4 Q14833 13/20 0.48
SGMS1 Q86VZ5 1/20 0.38
SGMS2 Q8NHU3 1/20 0.38
NPC1 O15118 2/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
FAAH O00519 1/20 0.36
CYP1A2 P05177 3/20 0.36
FADS1 O60427 1/20 0.36
CTSD P07339 1/20 0.36
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2235375 0.83 GRM4 (0.58) EPHX2GRM4SGMS1SGMS2NPC1
Hydrochloric Acid SCHEMBL2234357 0.82 GRM4 (0.56) EPHX2GRM4SGMS1SGMS2NPC1
SCHEMBL2234997 0.80 EPHX2 (0.60) EPHX2GRM4CYP1A2
SCHEMBL2236658 0.79 EPHX2 (0.60) EPHX2GRM4
SCHEMBL6923443 0.78 EPHX2 (0.69) EPHX2GRM4SGMS1SGMS2HPGD
SCHEMBL6923970 0.77 GRM4 (0.60) EPHX2GRM4NPC1RAB9ACYP1A2
SCHEMBL6922842 0.77 EPHX2 (0.64) EPHX2GRM4CYP1A2
SCHEMBL14804992 0.76 GRM4 (0.59) EPHX2GRM4NPC1HTTRAB9A
SCHEMBL6922687 0.76 EPHX2 (0.56) EPHX2GRM4CYP1A2
SCHEMBL14804987 0.74 GRM4 (0.56) EPHX2GRM4SGMS2HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011100614-A1 BENZISOXAZOLES AND AZABENZISOXAZOLES AS mgluR4 ALLOSTERIC POTENTIATORS, COMPOSITIONS, AND METHODS OF TREATING NEUROLOGICAL DYSFUNCTION VANDERBILT UNIVERSITY (US) 2011-08-18 WO disclosed