SCHEMBL6923762

SCHEMBL6923762

FC(F)(F)c1cc(Nc2noc3cccnc23)ccc1Cl

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.66
GRM4 Q14833 6/20 0.50
KDR P35968 2/20 0.43
PDGFRB P09619 1/20 0.43
KIT P10721 1/20 0.43
FLT1 P17948 1/20 0.43
ARNT P27540 1/20 0.43
EPAS1 Q99814 1/20 0.43
RAPGEF4 Q8WZA2 2/20 0.42
CYP1A2 P05177 1/20 0.42
RAPGEF3 O95398 2/20 0.41
CDK4 P11802 1/20 0.41
CDK2 P24941 1/20 0.41
BRAF P15056 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6922789 0.87 EPHX2 (0.67) EPHX2GRM4KDRKITCYP1A2
SCHEMBL14804991 0.86 EPHX2 (0.66) EPHX2GRM4KDRFLT1CYP1A2
SCHEMBL2234997 0.85 EPHX2 (0.60) EPHX2GRM4CYP1A2MEN1KMT2A
SCHEMBL6923970 0.83 GRM4 (0.60) EPHX2GRM4CYP1A2MEN1KMT2A
SCHEMBL2236658 0.81 EPHX2 (0.60) EPHX2GRM4KDR
SCHEMBL6922687 0.79 EPHX2 (0.56) EPHX2GRM4CYP1A2
SCHEMBL14804992 0.79 GRM4 (0.59) EPHX2GRM4RAPGEF4CYP1A2MEN1
SCHEMBL2235274 0.79 EPHX2 (0.74) EPHX2GRM4CYP1A2MEN1ALDH1A1
SCHEMBL2235367 0.79 GRM4 (0.61) EPHX2GRM4KDRPDGFRBKIT
SCHEMBL2235375 0.78 GRM4 (0.58) EPHX2GRM4MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011100614-A1 BENZISOXAZOLES AND AZABENZISOXAZOLES AS mgluR4 ALLOSTERIC POTENTIATORS, COMPOSITIONS, AND METHODS OF TREATING NEUROLOGICAL DYSFUNCTION VANDERBILT UNIVERSITY (US) 2011-08-18 WO disclosed