SCHEMBL6925935

SCHEMBL6925935

CCN(CC)CCOc1cc(NC(=O)c2ccc(C3CCCCC3)cc2)ccc1OC

nearest known ligand 0.73

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 16/20 0.73
HDAC3 O15379 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
DEGS1 O15121 1/20 0.48
HTR2C P28335 1/20 0.48
HPGD P15428 1/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
TP53 P04637 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6923836 0.88 MCHR1 (0.93) MCHR1HTR2C
SCHEMBL6807586 0.84 MCHR1 (0.65) MCHR1HDAC3HDAC11HDAC8HDAC6
SCHEMBL6926140 0.84 MCHR1 (0.72) MCHR1HTR2CNPC1ALDH1A1TP53
SCHEMBL6925370 0.83 MCHR1 (0.71) MCHR1HTR2CNPC1ALDH1A1TP53
SCHEMBL6923988 0.83 MCHR1 (0.71) MCHR1HTR2CNPC1ALDH1A1TP53
SCHEMBL6924087 0.83 MCHR1 (0.54) MCHR1HDAC3HDAC11HDAC8HDAC6
SCHEMBL6928256 0.82 MCHR1 (0.70) MCHR1HTR2CHPGDNPC1ALDH1A1
SCHEMBL6921439 0.81 MCHR1 (0.78) MCHR1HTR2CHPGDNPC1ALDH1A1
SCHEMBL6925692 0.81 MCHR1 (0.92) MCHR1HTR2C
SCHEMBL6927209 0.81 MCHR1 (0.78) MCHR1HTR2CHPGDNPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6515027-B1 Ligands, agonists or antagonists, of the CC chemokine receptor CC-CKR5 SMITHKLINE BEECHAM CORP. 2003-02-04 US disclosed
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed