SCHEMBL6926161

SCHEMBL6926161

COc1ccc(C(=O)Nc2ccc(OC)c(OCCN(C(C)C)C(C)C)c2)cc1

nearest known ligand 0.76

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 18/20 0.76
HTR2C P28335 1/20 0.73
NPC1 O15118 1/20 0.66
ALDH1A1 P00352 1/20 0.66
TP53 P04637 1/20 0.66
RAB9A P51151 1/20 0.66
SMN1; SMN2 Q16637 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6895261 0.91 MCHR1 (0.93) MCHR1HTR2C
SCHEMBL6920748 0.90 MCHR1 (0.71) MCHR1HTR2CNPC1ALDH1A1TP53
SCHEMBL6572097 0.90 MCHR1 (0.71) MCHR1HTR2CNPC1ALDH1A1TP53
SCHEMBL6926745 0.90 MCHR1 (0.71) MCHR1HTR2CNPC1ALDH1A1TP53
SCHEMBL6925443 0.90 MCHR1 (0.81) MCHR1HTR2C
Iodomethane SCHEMBL6899429 0.89 MCHR1 (0.89) MCHR1HTR2C
SCHEMBL6923778 0.89 MCHR1 (0.78) MCHR1HTR2C
SCHEMBL6926340 0.89 MCHR1 (0.92) MCHR1HTR2C
SCHEMBL6898082 0.89 MCHR1 (0.78) MCHR1HTR2C
SCHEMBL6896984 0.89 MCHR1 (0.78) MCHR1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6515027-B1 Ligands, agonists or antagonists, of the CC chemokine receptor CC-CKR5 SMITHKLINE BEECHAM CORP. 2003-02-04 US disclosed
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed