SCHEMBL6927975

SCHEMBL6927975

O=Cc1cc(-c2ccco2)ccc1F

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 6/20 0.70
KAT6A Q92794 1/20 0.42
PGR P06401 1/20 0.42
TAAR1 Q96RJ0 2/20 0.42
KEAP1 Q14145 1/20 0.41
PIK3R1 P27986 1/20 0.40
PIK3CA P42336 1/20 0.40
TDP2 O95551 2/20 0.38
FLT3 P36888 1/20 0.38
PTGES2 Q9H7Z7 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12767014 0.83 ERN1 (1.00) ERN1
SCHEMBL12767867 0.80 ERN1 (1.00) ERN1KEAP1
SCHEMBL28269364 0.78 ERN1 (0.54) ERN1KAT6APGRTAAR1KEAP1
SCHEMBL12121599 0.77 ERN1 (0.62) ERN1PGRTAAR1KEAP1PIK3R1
SCHEMBL15009764 0.77 ERN1 (0.77) ERN1PGRTAAR1KEAP1PIK3R1
SCHEMBL4036698 0.76 ERN1 (0.68) ERN1KEAP1PIK3R1PIK3CA
SCHEMBL20462888 0.74 ERN1 (0.46) ERN1KAT6APGRTAAR1KEAP1
SCHEMBL1125758 0.73 ERN1 (0.50) ERN1
SCHEMBL4037959 0.73 ERN1 (0.49) ERN1PIK3R1PIK3CACYP3A4
SCHEMBL9901972 0.72 ERN1 (0.50) ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518268-B1 Telomerase inhibitors and methods of their use GERON CORPORATION 2003-02-11 US disclosed
CN-1321153-A telomerase inhibitors and methods of use thereof GERON CORP (US) 2001-11-07 CN disclosed
WO-2001002377-A9 TELOMERASE INHIBITORS AND METHODS OF THEIR USE GERON CORP (US) 2001-10-11 WO disclosed
EP-1109796-A1 TELOMERASE INHIBITORS AND METHODS OF THEIR USE Geron Corporation (US) 2001-06-27 EP disclosed
WO-2001002377-A1 TELOMERASE INHIBITORS AND METHODS OF THEIR USE GERON CORPORATION (US) 2001-01-11 WO disclosed