SCHEMBL6928199

SCHEMBL6928199

Cn1c(-c2ccc(Cl)cc2)c(CCC(=O)Cl)c2cc(Cl)ccc21

nearest known ligand 0.65

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.65
TBXAS1 P24557 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6926561 0.90 TACR1 (0.65) TACR1TBXAS1
Hydrochloric Acid SCHEMBL7790354 0.89 TACR1 (0.64) TACR1TBXAS1
SCHEMBL7790361 0.86 TACR1 (0.61) TACR1
SCHEMBL6924338 0.81 TACR1 (0.75) TACR1
SCHEMBL7790320 0.81 TACR1 (0.54) TACR1TBXAS1
SCHEMBL7797019 0.80 TACR1 (0.55) TACR1TBXAS1
Hydrochloric Acid SCHEMBL7798859 0.79 TACR1 (0.53) TACR1TBXAS1
SCHEMBL7798879 0.78 TACR1 (0.52) TACR1TBXAS1
SCHEMBL7797108 0.78 TACR1 (0.57) TACR1
SCHEMBL7797105 0.78 TACR1 (0.57) TACR1TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518273-B1 2-aryl indole derivative as antagonists of tachykinins MERCK SHARP & DOHME LTD. 2003-02-11 US disclosed
WO-2000051984-A1 2-ARYL INDOLE DERIVATIVES AS ANTAGONISTS OF TACHYKININS MERCK SHARP & DOHME LIMITED (GB) 2000-09-08 WO disclosed