SCHEMBL6929688

SCHEMBL6929688

NC(Cc1ccccc1)C(O)C(O)C(N)Cc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.58
SLC15A1 P46059 1/20 0.55
SLC6A2 P23975 2/20 0.54
TAAR1 Q96RJ0 2/20 0.54
MAOA P21397 1/20 0.54
SLC6A4 P31645 1/20 0.54
SLC6A3 Q01959 1/20 0.54
SIGMAR1 Q99720 1/20 0.54
CYP2A6 P11509 1/20 0.54
ADORA2A P29274 1/20 0.54
ADORA1 P30542 1/20 0.54
ALPI P09923 1/20 0.54
PKM P14618 1/20 0.54
PTGS1 P23219 1/20 0.54
XIAP P98170 1/20 0.54
SLC7A5 Q01650 1/20 0.54
CSNK1E P49674 1/20 0.53
LAP3 P28838 3/20 0.50
ANPEP P15144 2/20 0.50
CYP2D6 P10635 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8482921 1.00 EPHX1 (0.58) EPHX1SLC15A1SLC6A2TAAR1MAOA
SCHEMBL14719648 1.00 EPHX1 (0.58) EPHX1SLC15A1SLC6A2TAAR1MAOA
SCHEMBL6931887 1.00 EPHX1 (0.58) EPHX1SLC15A1SLC6A2TAAR1MAOA
SCHEMBL6446300 1.00 EPHX1 (0.58) EPHX1SLC15A1SLC6A2TAAR1MAOA
SCHEMBL9740410 1.00 EPHX1 (0.58) EPHX1SLC15A1SLC6A2TAAR1MAOA
SCHEMBL6445044 1.00 EPHX1 (0.58) EPHX1SLC15A1SLC6A2TAAR1MAOA
SCHEMBL7144488 1.00 EPHX1 (0.58) EPHX1SLC15A1SLC6A2TAAR1MAOA
SCHEMBL7190709 1.00 EPHX1 (0.58) EPHX1SLC15A1SLC6A2TAAR1MAOA
SCHEMBL6446370 1.00 EPHX1 (0.58) EPHX1SLC15A1SLC6A2TAAR1MAOA
SCHEMBL7168775 1.00 EPHX1 (0.58) EPHX1SLC15A1SLC6A2TAAR1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0801640-B1 2,5-DIAMINO-3,4-DISUBSTITUTED-1,6-DIPHENYLHEXANE ISOSTERES COMPRISING BENZAMIDE, SULFONAMIDE AND ANTHRANILAMIDE SUBUNITS AND METHODS OF USING SAME USA (US) 2003-03-26 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
EP-0674513-A4 1995-10-25 EP disclosed
EP-0674513-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS. ABBOTT LAB (US) 1995-10-04 EP disclosed
EP-0665215-A1 1,4-Diamino-2,3-dihydroxybutanes THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-08-02 EP disclosed
US-5430155-A Viricides, treatment of AIDS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-07-04 US disclosed
WO-1994014436-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1994-07-07 WO disclosed
US-5294720-A Viricides THE DUPONT MERCK PHARMACEUTICAL CO. (US) 1994-03-15 US disclosed
EP-0532693-A1 1,4-DIAMINO-2,3-DIHYDROXYBUTANES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-03-24 EP disclosed
WO-1991018866-A2 1,4-DIAMINO-2,3-DIHYDROXYBUTANES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-12-12 WO disclosed