SCHEMBL6929861

SCHEMBL6929861

CC(C)(C)CCNC(=O)c1cnc(OCc2cccc(F)c2)c(N)c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.48
MAOB P27338 3/20 0.42
PARP10 Q53GL7 1/20 0.42
PDGFRB P09619 1/20 0.41
KDR P35968 1/20 0.41
NR4A2 P43354 2/20 0.40
SGMS2 Q8NHU3 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.40
CHRM4 P08173 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6928898 0.89 GRM5 (0.48) GRM5MAOBPARP10NR4A2SGMS2
SCHEMBL6929584 0.87 GRM5 (0.47) GRM5MAOBSGMS2MRGPRX4
SCHEMBL6927929 0.86 GRM5 (0.46) GRM5MAOBNR4A2SGMS2MRGPRX4
SCHEMBL2158904 0.83 GRM5 (0.68) GRM5MAOB
SCHEMBL6929950 0.76 GRM5 (0.54) GRM5MAOBPARP10NR4A2SGMS2
SCHEMBL6929270 0.74 GRM5 (0.47) GRM5MAOBMRGPRX4
SCHEMBL6931129 0.73 GRM5 (0.51) GRM5MAOB
SCHEMBL6929241 0.73 GRM5 (0.55) GRM5
SCHEMBL9990257 0.73 MRGPRX4 (0.44) GRM5NR4A2MRGPRX4
SCHEMBL6930489 0.72 MEN1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011035324-A1 O-BENZYL NICOTINAMIDE ANALOGS AS MGLUR5 POSITIVE ALLOSTERIC MODULATORS VANDERBILT UNIVERSITY (US) 2011-03-24 WO disclosed