SCHEMBL6933368

SCHEMBL6933368

NC(=O)c1ccc(CCCO)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 2/20 0.59
CA2 P00918 3/20 0.53
CYP4F2 P78329 1/20 0.53
PLA2G10 O15496 1/20 0.52
PLA2G2A P14555 1/20 0.52
PARP10 Q53GL7 4/20 0.48
PPARA Q07869 1/20 0.45
CYP17A1 P05093 1/20 0.44
DPP4 P27487 4/20 0.44
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
PARP15 Q460N3 1/20 0.43
PARP14 Q460N5 1/20 0.43
PARP16 Q8N5Y8 1/20 0.43
PARP11 Q9NR21 1/20 0.43
PARP4 Q9UKK3 1/20 0.43
HSD17B10 Q99714 2/20 0.43
POLB P06746 1/20 0.43
CYP3A4 P08684 1/20 0.43
PARP1 P09874 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10622023 0.98 CYP4A11 (0.58) CYP4A11CA2CYP4F2PLA2G10PLA2G2A
SCHEMBL9761155 0.94 CYP4A11 (0.61) CYP4A11CA2CYP4F2PLA2G10PLA2G2A
SCHEMBL8684163 0.89 CYP4A11 (0.58) CYP4A11CA2CYP4F2PLA2G10PLA2G2A
SCHEMBL2633786 0.87 PLA2G10 (0.55) CYP4A11CA2CYP4F2PLA2G10PLA2G2A
SCHEMBL4037830 0.83 PLA2G10 (0.52) PLA2G10PLA2G2APARP10CYP17A1ALDH1A1
SCHEMBL13686091 0.83 CYP4A11 (0.63) CYP4A11CA2CYP4F2PPARAHSD17B10
SCHEMBL7028830 0.83 CYP4A11 (0.63) CYP4A11CA2CYP4F2PPARAHSD17B10
SCHEMBL5330371 0.82 PLA2G10 (0.50) CYP4A11PLA2G10PLA2G2APARP10CYP17A1
SCHEMBL9101894 0.82 PARP10 (0.55) CA2PLA2G10PLA2G2APARP10DPP4
SCHEMBL29222811 0.82 PLA2G10 (0.50) CYP4A11PLA2G10PLA2G2APARP10CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101993416-A Quinoline compound and preparation method thereof, medicament combination containing compound and application of compound SHANGHAI INST MATERIA MEDICA 2011-03-30 CN claimed
CN-101993416-B Quinoline compound and preparation method thereof, medicament combination containing compound and application of compound SHANGHAI INST MATERIA MEDICA 2013-09-11 CN disclosed
CN-101993416-A Quinoline compound and preparation method thereof, medicament combination containing compound and application of compound SHANGHAI INST MATERIA MEDICA 2011-03-30 CN disclosed
EP-0768307-B1 Heterocyclic tertiary amines, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-11-26 EP disclosed
EP-0768307-A1 Heterocyclic tertiary amines, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1997-04-16 EP disclosed