SCHEMBL6943766

SCHEMBL6943766

CC(C)Oc1c(CNc2ccccn2)cc(Cc2ccccc2)cc1C(=O)CC(=O)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP1 P07148 1/20 0.39
FABP6 P51161 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ALDH1A1 P00352 4/20 0.37
HPGD P15428 1/20 0.37
BDKRB1 P46663 1/20 0.35
POLB P06746 1/20 0.35
ITGB3 P05106 2/20 0.35
ITGAV P06756 2/20 0.35
ITGB1 P05556 1/20 0.35
ITGB5 P18084 1/20 0.35
ITGB6 P18564 1/20 0.35
CXCR4 P61073 1/20 0.35
GAA P10253 2/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PTPN1 P18031 2/20 0.34
PTPN2 P17706 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947887 0.79 PTPN1 (0.38) L3MBTL1ALDH1A1HPGDPTPN1PTPN2
SCHEMBL6943763 0.79 ERCC5 (0.34) L3MBTL1ALDH1A1MAPTPTPN1LMNA
SCHEMBL6951272 0.78 KDM4E (0.43) ALDH1A1PTPN1PTPN2PTPN6LMNA
SCHEMBL7074788 0.77 CYP19A1 (0.39) PTPN1PTPN2PTPN6
SCHEMBL6947879 0.77 ERCC5 (0.41) L3MBTL1MAPTPTPN1PTPN2PTPN6
SCHEMBL6948187 0.76 ERCC5 (0.40) L3MBTL1ALDH1A1HPGDGAAMAPT
SCHEMBL6948110 0.76 MEN1 (0.44) ALDH1A1HPGDPOLBMEN1KMT2A
Dimethylamine SCHEMBL6949345 0.75 SMN1; SMN2 (0.41) L3MBTL1NPSR1ALDH1A1HPGDPOLB
SCHEMBL7077955 0.75 CYP19A1 (0.39) MEN1KMT2ALMNA
SCHEMBL6950058 0.75 ERCC5 (0.39) ALDH1A1PTPN1PTPN2PTPN6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed