SCHEMBL6945818

SCHEMBL6945818

Cn1c(=O)[nH]c2nc(N3CCNCC3)n(-c3ccccc3Cl)c2c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 5/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ADRB1 P08588 2/20 0.46
POLB P06746 1/20 0.41
SIRT5 Q9NXA8 1/20 0.41
ALDH1A1 P00352 3/20 0.39
KDM4C Q9H3R0 1/20 0.39
HTR2C P28335 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
RAB9A P51151 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
HSD17B10 Q99714 1/20 0.38
DRD2 P14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5718931 0.92 DPP4 (0.42) DPP4L3MBTL1ADRB1POLBSIRT5
SCHEMBL5792690 0.83 DPP4 (0.64) DPP4L3MBTL1POLBSIRT5ALDH1A1
SCHEMBL27623297 0.82 DPP4 (0.49) DPP4L3MBTL1ADRB1POLBSIRT5
SCHEMBL5719678 0.82 DPP4 (0.68) DPP4L3MBTL1ADRB1ALDH1A1KMT2A
SCHEMBL2954897 0.81 GAA (0.44) L3MBTL1MEN1KMT2AMAPTGAA
Trifluoroacetic Acid SCHEMBL5719494 0.76 DPP4 (0.58) DPP4L3MBTL1POLBSIRT5ALDH1A1
SCHEMBL13200001 0.76 DPP4 (0.44) DPP4L3MBTL1ADRB1ALDH1A1HTR2C
SCHEMBL5789362 0.75 DPP4 (0.61) DPP4L3MBTL1ADRB1ALDH1A1HTR2C
SCHEMBL5792563 0.75 DPP4 (0.56) DPP4L3MBTL1ALDH1A1TSHR
Trifluoroacetic Acid SCHEMBL2954275 0.73 DPP4 (0.42) DPP4L3MBTL1ADRB1ALDH1A1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1338595-A2 Xanthine derivatives as DPP-IV inhibitors Eisai Co., Ltd. (JP) 2003-08-27 EP disclosed