SCHEMBL6946145

SCHEMBL6946145

NCc1cccc2ccccc12.O=C(N[C@@H](CCCNC1CCCc2cccnc21)C(=O)O)c1ccc(CNc2ccccn2)c2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
CXCR4 P61073 6/20 0.35
FOLH1 Q04609 1/20 0.34
ADORA2A P29274 1/20 0.34
FNTA P49354 3/20 0.33
FNTB P49356 3/20 0.33
ITGAV P06756 2/20 0.33
ITGB3 P05106 1/20 0.33
PGGT1B P53609 1/20 0.33
ITGB6 P18564 1/20 0.32
SLC40A1 Q9NP59 1/20 0.32
CASR P41180 1/20 0.32
CTSL P07711 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7150127 0.94 HDAC1 (0.42) HDAC1HDAC6CXCR4FOLH1ADORA2A
SCHEMBL6990541 0.91 FOLH1 (0.37) HDAC1HDAC6CXCR4FOLH1ADORA2A
SCHEMBL6018818 0.91 FOLH1 (0.37) HDAC1HDAC6CXCR4FOLH1ADORA2A
SCHEMBL6018347 0.91 FOLH1 (0.37) HDAC1HDAC6CXCR4FOLH1ADORA2A
SCHEMBL6018408 0.90 HDAC1 (0.38) HDAC1HDAC6CXCR4ADORA2AITGAV
SCHEMBL6681750 0.83 HDAC1 (0.54) HDAC1HDAC6CXCR4FOLH1ADORA2A
SCHEMBL6018112 0.83 HDAC1 (0.44) HDAC1HDAC6CXCR4ADORA2ASLC40A1
SCHEMBL6018467 0.83 CXCR4 (0.36) HDAC1HDAC6CXCR4ADORA2AFNTA
SCHEMBL6018159 0.83 HDAC1 (0.41) HDAC1HDAC6CXCR4ADORA2AFNTA
SCHEMBL7150122 0.82 HDAC1 (0.42) HDAC1HDAC6CXCR4FOLH1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound KUREHA CORPORATION (JP) 2004-08-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound CXCR4, CXCR1, CXCR2 HDAC1 1092/4885HDAC6 1799/4885CXCR4 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.