SCHEMBL6948666

SCHEMBL6948666

NCCON=C(CCCN1CCC(C(=O)c2ccccc2)CC1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.54
HTR2A P28223 2/20 0.51
HRH2 P25021 1/20 0.48
HRH1 P35367 1/20 0.48
KDM4E B2RXH2 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
HRH3 Q9Y5N1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6948664 1.00 KCNH2 (0.54) KCNH2HTR2AHRH2HRH1KDM4E
SCHEMBL6947200 0.94 HTR2A (0.57) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL6947854 0.94 HTR2A (0.57) KCNH2HTR2AKDM4ECYP1A2CYP3A4
Hydrochloric Acid SCHEMBL8867634 0.93 HTR2A (0.56) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8867625 0.93 HTR2A (0.56) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL6952317 0.92 HRH2 (0.49) KCNH2HTR2AHRH2HRH1HRH3
SCHEMBL6952321 0.92 HRH2 (0.49) KCNH2HTR2AHRH2HRH1HRH3
SCHEMBL6947026 0.92 MEN1 (0.53) KCNH2HTR2AHRH2HRH1KDM4E
SCHEMBL6947024 0.92 MEN1 (0.53) KCNH2HTR2AHRH2HRH1KDM4E
SCHEMBL6953050 0.91 HTR2A (0.53) HTR2AKDM4ECYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709378-B1 Aminoalkyloximes, a process for their preparation, their use as medicaments and intermediate compounds AVENTIS PHARMA INC (US) 2003-03-19 EP disclosed
US-5665756-A Aminoalkyloximes useful in the treatment of depression and obsessive compulsive disorders HOECHST MARION ROUSSEL, INC. (US) 1997-09-09 US disclosed
US-5648367-A ANTIDEPRESANTS, OBSESSIVE-COMPULSIVE DISORDER HOECHST MARION ROUSSEL, INC. (US) 1997-07-15 US disclosed
EP-0709378-A2 Aminoalkyloximes, a process for their preparation, their use as medicaments and intermediate compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1996-05-01 EP disclosed