SCHEMBL6949689

SCHEMBL6949689

CCNC1CN(c2c(F)cc3c(=O)c(OC(=O)O)cn(-c4nc(N)c(F)cc4F)c3c2Br)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.51
CYP3A4 P08684 2/20 0.51
TOP1 P11387 3/20 0.33
KCNH2 Q12809 4/20 0.33
KDM4E B2RXH2 4/20 0.32
HPGD P15428 4/20 0.32
ALDH1A1 P00352 3/20 0.32
HSD17B10 Q99714 3/20 0.32
PMP22 Q01453 1/20 0.32
CYP2C19 P33261 1/20 0.31
LMNA P02545 2/20 0.31
POLB P06746 1/20 0.31
XBP1 P17861 1/20 0.31
NFKB1 P19838 1/20 0.31
HTT P42858 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
HRH3 Q9Y5N1 2/20 0.31
TOP2A P11388 5/20 0.30
TOP2B Q02880 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7861212 0.91 CYP3A4 (0.53) CYP2C9CYP3A4TOP1KCNH2KDM4E
SCHEMBL2912243 0.91 CYP2C9 (0.62) CYP2C9CYP3A4TOP1KCNH2KDM4E
Fumaric Acid SCHEMBL2922599 0.87 CYP2C9 (0.58) CYP2C9CYP3A4TOP1KCNH2KDM4E
Maleic Acid SCHEMBL2922594 0.87 CYP2C9 (0.58) CYP2C9CYP3A4TOP1KCNH2KDM4E
SCHEMBL27462343 0.86 CYP3A4 (0.51) CYP2C9CYP3A4TOP1KCNH2KDM4E
SCHEMBL2921570 0.81 CYP3A4 (0.65) CYP2C9CYP3A4TOP1KCNH2KDM4E
SCHEMBL2920475 0.81 CYP3A4 (0.52) CYP2C9CYP3A4TOP1KCNH2KDM4E
SCHEMBL6281366 0.81 CYP2C9 (0.77) CYP2C9CYP3A4TOP1KCNH2KDM4E
SCHEMBL2918028 0.81 CYP3A4 (0.62) CYP2C9CYP3A4TOP1KCNH2KDM4E
Hydrochloric Acid SCHEMBL2923148 0.80 CYP3A4 (0.62) CYP2C9CYP3A4TOP1KCNH2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1193266-B1 QUINOLINECARBOXYLIC ACID DERIVATIVE OR SALTS THEREOF WAKUNAGA PHARMA CO LTD (JP) 2003-08-27 EP claimed