SCHEMBL6953754

SCHEMBL6953754

O=C(O)C(OCC1(c2ccc(N3CCC(c4ccc(F)cc4)CC3)cc2)CCCCC1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.54
KCNH2 Q12809 2/20 0.43
FAAH O00519 1/20 0.40
CCR2 P41597 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6952152 0.83 TACR1 (0.68) TACR1KCNH2FAAHCCR2
SCHEMBL6494295 0.83 TACR1 (0.78) TACR1KCNH2CCR2
SCHEMBL6965411 0.78 TACR1 (0.57) TACR1KCNH2CCR2
SCHEMBL6485287 0.75 TACR1 (0.66) TACR1KCNH2CCR2
SCHEMBL7163593 0.74 TACR1 (0.49) TACR1KCNH2FAAHCCR2
SCHEMBL7000788 0.73 TACR1 (0.68) TACR1KCNH2CCR2
SCHEMBL6960087 0.71 CYP3A4 (0.48) TACR1FAAH
SCHEMBL6483284 0.71 TACR1 (0.72) TACR1KCNH2CCR2
Hydrochloric Acid SCHEMBL6963690 0.70 CYP3A4 (0.47) FAAH
SCHEMBL6484641 0.70 TACR1 (1.00) TACR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286978-A1 CYCLOHEXYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 2003-03-05 EP disclosed
WO-2001087866-A1 CYCLOHEXYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 2001-11-22 WO disclosed