SCHEMBL6957201

SCHEMBL6957201

COC(=O)CC(=O)CC(O)/C=C/c1c(C(C)C)cc(C)nc1-c1ccc(F)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 3/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
PDE6D O43924 1/20 0.41
NR1I2 O75469 1/20 0.41
PDE4D Q08499 1/20 0.41
ESR1 P03372 1/20 0.40
CHRM1 P11229 1/20 0.40
TBXA2R P21731 1/20 0.40
PDE4A P27815 1/20 0.40
ADRA1A P35348 1/20 0.40
ABCC3 O15438 1/20 0.40
ABCC4 O15439 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27530291 0.91 HMGCR (0.33) HMGCRHDAC1HDAC2HDAC6ALDH1A1
SCHEMBL9261685 0.90 HMGCR (0.46) HMGCRHDAC1HDAC2HDAC6ALDH1A1
SCHEMBL9261677 0.90 HMGCR (0.46) HMGCRHDAC1HDAC2HDAC6ALDH1A1
SCHEMBL6962901 0.83 HMGCR (0.49) HMGCRHDAC1HDAC2HDAC6ALDH1A1
SCHEMBL10517235 0.82 HMGCR (0.40) HMGCRHDAC1HDAC2HDAC6ALDH1A1
SCHEMBL27312221 0.82 HMGCR (0.44) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL6961463 0.79 HMGCR (0.39) HMGCRHDAC1HDAC2HDAC6ALDH1A1
SCHEMBL8949894 0.79 HMGCR (0.58) HMGCRHDAC1HDAC2HDAC6ALDH1A1
SCHEMBL8949666 0.79 HMGCR (0.44) HMGCRNR1I2PDE4DESR1CHRM1
SCHEMBL6957249 0.79 HMGCR (0.46) HMGCRHDAC1HDAC2HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325130-B1 Substituted pyridines BAYER AG (DE) 2003-11-05 EP disclosed
EP-1123924-A1 Substituted pyridines as HMG-COA reductase inhibitors BAYER AG (DE) 2001-08-16 EP disclosed
EP-1123925-A1 Process for preparation of substituted pyridines BAYER AG (DE) 2001-08-16 EP disclosed
CN-1055684-C Process for preparing substituted pyridine compounds BAYER AG (DE) 2000-08-23 CN disclosed
CN-1034364-A Substituted pyridines and process for their preparation BAYER AG (DE) 1989-08-02 CN disclosed
EP-0325130-A2 Substituted pyridines BAYER AG (DE) 1989-07-26 EP disclosed