SCHEMBL6961876

SCHEMBL6961876

Clc1ccccc1-c1[nH]nc2c1CCc1ccccc1-2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.50
GSR P00390 2/20 0.50
HTR7 P34969 1/20 0.50
DRD4 P21917 1/20 0.48
KDR P35968 2/20 0.47
RAB9A P51151 3/20 0.46
DCUN1D1 Q96GG9 1/20 0.45
CDK1 P06493 1/20 0.43
CDK2 P24941 1/20 0.43
CHEK1 O14757 1/20 0.42
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
ALPL P05186 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969848 0.82 NPC1 (0.48) NPC1GSRHTR7DRD4KDR
SCHEMBL11865968 0.82 NPC1 (0.53) NPC1GSRHTR7KDRRAB9A
SCHEMBL11861088 0.81 KDR (0.56) NPC1GSRHTR7KDRRAB9A
SCHEMBL6965340 0.79 NPC1 (0.48) NPC1GSRHTR7DRD4KDR
SCHEMBL12567897 0.78 KDR (0.74) NPC1GSRHTR7DRD4KDR
SCHEMBL8063320 0.78 NPC1 (0.65) NPC1GSRKDRRAB9ACDK1
SCHEMBL11839656 0.77 NPC1 (0.51) NPC1GSRHTR7KDRRAB9A
SCHEMBL6968969 0.77 NPC1 (0.48) NPC1GSRKDRRAB9ACDK1
SCHEMBL11863189 0.77 GSR (0.48) NPC1GSRKDRRAB9ACDK1
Methane SCHEMBL8064257 0.77 NPC1 (0.64) NPC1GSRKDRRAB9ACDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023063-B1 INDENO[1,2-c], NAPHTHO[1,2-c]- AND BENZO[6,7]CYCLOHEPTA[1,2-c]PYRAZOLE DERIVATIVES ABBOTT GMBH & CO KG (DE) 2003-09-10 EP disclosed
US-6451834-B1 Indeno[1,2-c]-, naphtho[1,2-c]- and benzo[6,7]cyclohepta[1,2-c]pyrazole derivatives BASF AKTIENGESELLSCHAFT (DE) 2002-09-17 US disclosed
EP-1023063-A1 INDENO 1,2-c]-, NAPHTHO 1,2-c]- AND BENZO 6,7]CYCLOHEPTA 1,2-c]PYRAZOLE DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 2000-08-02 EP disclosed
WO-1999017769-A1 INDENO[1,2-c]-, NAPHTHO[1,2-c]- AND BENZO[6,7]CYCLOHEPTA[1,2-c]PYRAZOLE DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 1999-04-15 WO disclosed